The first synthesis and cytostatic activity of novel 6-(fluoromethyl)purine bases and nucleosides.

نویسندگان

  • Peter Silhár
  • Radek Pohl
  • Ivan Votruba
  • Michal Hocek
چکیده

Two alternative approaches to the synthesis of novel 6-(fluoromethyl)purine bases and nucleosides are described either by direct deoxyfluorination or by multistep functional group transformations starting from 6-(hydroxymethyl)purines. 6-(fluoromethyl)purine ribonucleoside displayed significant cytostatic effects.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 3 16  شماره 

صفحات  -

تاریخ انتشار 2005